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. 2025 Aug 22;5:367. doi: 10.1038/s43856-025-01033-z

Table 1.

Binding of [68Ga]Ga-DOTA-mDesmo to purified human V1b receptor

Binding (%) (Mean ± SD)
V1b (15.6 nM) + [68Ga]Ga-DOTA-mDesmo 5.1 ± 1.3
V1b (31. 25 nM) + [68Ga]Ga-DOTA-mDesmo 21.8 ± 2.1
V1b (62.5 nM) + [68Ga]Ga-DOTA-mDesmo 25.7 ± 2.4
V1b (125 nM) + [68Ga]Ga-DOTA-mDesmo 30.7 ± 1.9
V1b (250 nM) + [68Ga]Ga-DOTA-mDesmo 44 ± 2.2
V1b (250 nM) + [68Ga]Ga-DOTA-mDesmo + DOTA-mDesmo (5 µM) 38.8 ± 1.7
V1b (250 nM) + [68Ga]Ga-DOTA-mDesmo + DOTA-mDesmo (20 µM) 22.1 ± 2.1