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. 2025 Aug 22;16:7854. doi: 10.1038/s41467-025-62288-7

Table 1.

The kinetic parameters of Bufalin and ESR1, CYP17A1, and PKC delta binding from SPRi

Protein Avg ka (1/Ms) Avg kd (1/s) Avg KD (M) ABS (tr_KD)
ESR1 1.29E + 02 6.98E−04 5.42E−06 17.492
CYP17A1 2.50E + 00 7.36E−02 2.94E−02 5.086
PKC delta 1.79E + 01 2.31E−01 1.29E−02 6.271