Skip to main content
. 2025 Jul 28;16(11):3537–3550. doi: 10.7150/jca.118273

Table 2.

Occurrence and Potential treatment of H3K14-related diseases

The name of the disease Mechanism of impact Potential therapeutic targets/measures Reference
Cutaneous T Cell Lymphoma (CTCL) Genome-wide H3K9/14ac (H3ac) and H3K27ac levels were significantly increased HDACi 97
Renal Cell Carcinoma (RCC) Renal oxidative stress, high DNA methylation, low H3 acetylation Raise the level of oxidative stress 98
Acute promyelocytic leukemia (APL) The PML-RARA fusion protein recruits HDAC/HMT to form an inhibitory complex that blocks differentiation gene expression. Belinostat and 3-Deazaneplanocin A directly disrupt the complex and reverse the apparent silencing by H3K14ac elevation HDAC inhibitor combined with HMT inhibitor; EGCG 85, 99
Breast cancer Increased expression of ATP-binding cassette (ABC)
-type transporters
RNAi down-regulated the expression of HATs PCAF and GCN5 100
Abdominal Aortic Aneurysm (AAA) There is increased acetylation of H3K14 and DNA
hypomethylation
mRNA levels of DNMT and HDAC 101, 102
Glioma IDH1 mutations can lead to a wide range of DNA and histone methylation; Overexpression of HCMV IE86 protein The joint HDACi cAMP agonist, ATF5expression 10, 103, 104
Nasopharyngeal carcinoma Upregulation of AFAP1-AS1, H3K14acetylation and protein binding to the brominated domain of TIF1α Enhanced KAT2Bacetyltransferase activation and YAP mRNA stabilization 31
Periodontitis Cut GCN5 activated PDLSCs Wnt/beta Catenin signaling pathway, H3K14ac level is low Up-regulation of GCN5 83, 105
Mastitis H3K14 high acetylation,
lipopolysaccharide
Metformin activates AMPK signaling pathway to reverse H3K14hyperacetylation 106-108
Acute necrotizing pancreatitis (AP) The key initiating cytokine TNF-AP was strongly up-regulated and H3K14 acetylation was increased 109
Asthma PMCS, increasethe CD4 + T cells inthe IL - 4 gene promoter H3K14 acetylation and H3K27me3 Notch Signaling pathway 20, 110
Diabetes SIRT2 expression was decreased, EPB41L4A-AS1 binding to GCN5, andH3K14 level was increased. Claudin-5 is deficient Upregulation of SIRT2; EPB41L4A-AS1; Ketoβ-hydroxybutyricacid (BHB) therapy 30, 61, 111, 112
Neurodegenerative disease Friedreich's ataxia FXN introns within the GAA x TTC triplets amplification result in transcriptional silencing, with histone H3 acetylation HDACi 53
Intrauterine growth retardation (IUGR) Prenatal caffeine exposure increased the mRNA expression of DNAmethyltransferases Dnmt1, Dnmt3a, HDAC1, and HDAC2, and decreased the acetylation level of H3K14 DNA methylation and histone acetylation 113, 114
Tuberculosis (TB) HDAC1 gene/protein expression increases, H3K14Ac decrease Downregulation of HDAC 115