Table 3. Cell viability of SH-SY5Y and HEK293 cells treated with the compounds for 24 h. Data are mean ± SD (n = 3).
| Compounds | IC50 (μM) | ||
|---|---|---|---|
| SH-SY5Y | HEK-293 | Selectivity | |
| 10a | 8.22 ± 0.12 | 78.21 ± 0.42 | 9.5 |
| 10b | 15.82 ± 0.20 | 43.42 ± 0.36 | 2.7 |
| 10c | 11.93 ± 0.20 | 46.91 ± 0.32 | 3.9 |
| 10d | 16.37 ± 0.21 | 75.22 ± 0.35 | 4.6 |
| 10e | 33.19 ± 0.25 | 68.95 ± 0.41 | 2.1 |
| 10f | 7.33 ± 0.11 | 33.18 ± 0.55 | 4.5 |
| 10g | 12.94 ± 0.13 | 86.45 ± 0.52 | 6.7 |
| 10h | 7.42 ± 0.07 | 78.38 ± 0.57 | 10.6 |
| 10i | 4.26 ± 0.08 | 37.39 ± 0.55 | 8.8 |
| 10j | 6.75 ± 0.18 | 67.43 ± 0.47 | 10.0 |
| 10k | 8.11 ± 0.07 | 81.71 ± 0.56 | 10.1 |
| 10l | 42.15 ± 0.37 | 92.86 ± 0.71 | 2.2 |
| 10m | 28.33 ± 0.26 | 46.45 ± 0.45 | 1.6 |
| 10n | 5.22 ± 0.12 | 38.42 ± 0.19 | 7.4 |
| Sorafenib | 3.88 ± 0.12 | 16.22 ± 0.14 | 4.2 |