Table 1. SAR exploration of the DHBA group.
| |||
|---|---|---|---|
| Cpd. | R1 | Linker | AXL IC50 (nM) |
| w0 |
|
|
17 |
| w1 |
|
|
26 |
| w2 |
|
|
34 |
| w3 |
|
|
>1000 |
| w4 |
|
|
14 |
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