Table 1.
Classes of reported bacterial fatty acid synthesis (FASII) inhibitors.
| Inhibitor Class | Target Bacteria | References |
|---|---|---|
| Diazaborines | E. coli, S. aureus | [68] |
| 1,2,3,4-tetrahydro-1H-pyrido [3,4-b]indole derivatives | S. aureus, Enterococcus faecalis | [69] |
| 1H-imidazole derivatives | S. aureus, E. coli | [70] |
| Diphenyl ethers and triclosan analogs | E. coli, M. tuberculosis | [71] |
| Naphthyridinones | S. aureus, S. pneumoniae | [69] |
| Acrylamide-based compounds | M. tuberculosis | [72] |
| 1,5,6,7-tetrahydroindeno [5,6-d]imidazoles | M. tuberculosis | [73] |
| Coumarin derivatives | M. tuberculosis, S. aureus | [74] |
| Pyrone/pyridone derivatives | M. tuberculosis | [75] |
| Pyrrolidine-based inhibitors | P. aeruginosa | [76] |
| Quinoline/quinoxaline derivatives | M. tuberculosis | [77] |
| N′-benzoylbenzohydrazides | M. tuberculosis | [78] |