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. 2025 Jul 27;18(8):1119. doi: 10.3390/ph18081119

Table 1.

Classes of reported bacterial fatty acid synthesis (FASII) inhibitors.

Inhibitor Class Target Bacteria References
Diazaborines E. coli, S. aureus [68]
1,2,3,4-tetrahydro-1H-pyrido [3,4-b]indole derivatives S. aureus, Enterococcus faecalis [69]
1H-imidazole derivatives S. aureus, E. coli [70]
Diphenyl ethers and triclosan analogs E. coli, M. tuberculosis [71]
Naphthyridinones S. aureus, S. pneumoniae [69]
Acrylamide-based compounds M. tuberculosis [72]
1,5,6,7-tetrahydroindeno [5,6-d]imidazoles M. tuberculosis [73]
Coumarin derivatives M. tuberculosis, S. aureus [74]
Pyrone/pyridone derivatives M. tuberculosis [75]
Pyrrolidine-based inhibitors P. aeruginosa [76]
Quinoline/quinoxaline derivatives M. tuberculosis [77]
N′-benzoylbenzohydrazides M. tuberculosis [78]