Table 1.
PDB ID and important amino acids involved in the interaction of GP63, FPPS, and NMT proteins with plant compounds.
| Protein name | Code PDB | Resolution | Amine acids | Reference No. |
|---|---|---|---|---|
| GP63 | 1LML | 1.86 Å | HIS264, HIS268, HIS334, MET345, ALA348, ALA227, SER273, GLY222, THR228, GLU265, ALA350, PRO347, VAL223, GLY329, GLU220 LEU224, ALA225, SER418, GLN341, GLY222, SER465, VAL223, HIS264, LEU257, PRO460, ALA350 HIS264, ASP342, HIS268, HIS334, MET345, ALA348, PHE272, SER333 |
(25) (26) (17) |
| FPPS | 4K10 | 2.30 A | LYS207, LYS264, ARG107, ASP102, ASP98, ASP99, ASP250, PHE94, LEU95, HIS93, MET101, GLN167 ARG107, GLN167, LYS264, ASP268, THR267, ASP170, LYS207 LYS207, LYS264, ARG107, PHE94, GLN167, THR163, ASP102, ASP98, ASP250, ASP254 ASP98, ILE100, MET101, ASP102, ARG107, ARG108, HIS93, PHE94 |
(27) (28) (19) (29) |
| NMT | 4CGO | 1.30 A | PHE90, VAL81, PHE232, GLY397, PHE88, HIS219, ASP83, GLY205, TYR80, TYR217, LEU421, TYR345, LEU341, TYR92, ASN167, HIS398, ALA204, VAL374, ALA343, ASN376 TYR92, PHE90, ASN167, PHE88, THR203, HIS219, TYR217, PHE232, TYR326, VAL81, TYR80, GLU82, ILE328, SER330, LEU341, MET420, LEU421, ASP396, LEU399, ASP396, ASN376, VAL374, TYR345, ALA343 ALA204, TYR202, PHE90, MET420, TYR326, TYR345, LEU421, ASN167, VAL81, ASN383, TYR80, VAL378, LYS173, GLU82 |
(9) (30) (31) |
GP63, Glycoprotein 63; FPPS, farnesyl diphosphate synthase; NMT, N-myristoyltransferase.