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. 2025 Aug 20;68(17):18407–18422. doi: 10.1021/acs.jmedchem.5c01160

3. Improvement in PK Parameters via Linker and CRBN Ligand Modification.

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*Racemic at 3-hydroxypiperidine. **Units of nM. @Units of mL/min/kg. $Units of 10–6 cm/s. #IV (2 mg/kg)/PO (10 mg/kg), Cl in units of mL/min/kg, Vss in units of L/kg, T 1/2 in units of h.