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. Author manuscript; available in PMC: 2025 Sep 21.
Published before final editing as: Crit Rev Biochem Mol Biol. 2025 Aug 22:1–34. doi: 10.1080/10409238.2025.2545785

Table 7.

Reported AOX inhibitors.

Compound Microorganism targeted IC50

Ascochlorin T. brucei brucei 3.7 nM (Young et al. 2020; Xu et al. 2021)
Ascofuranone T. brucei brucei 0.03 nM (Shiba et al. 2013)
Octyl gallate T. brucei brucei 0.23 μM (Young et al. 2020)
Salicylhydroxamic acid (SHAM) T. brucei brucei 6 μM (Meco-Navas et al. 2018)
Salicylic hydroxamic acid T. brucei brucei 4 nM (Young et al. 2020)
8-Hydroxyquinoline P. falciparum 11 μM (Roberts et al. 2004)
8-Hydroxyquinoline C. parvum 0.7 μM (Roberts et al. 2004)