Table 7.
Reported AOX inhibitors.
Compound | Microorganism targeted | IC50 |
---|---|---|
| ||
Ascochlorin | T. brucei brucei | 3.7 nM (Young et al. 2020; Xu et al. 2021) |
Ascofuranone | T. brucei brucei | 0.03 nM (Shiba et al. 2013) |
Octyl gallate | T. brucei brucei | 0.23 μM (Young et al. 2020) |
Salicylhydroxamic acid (SHAM) | T. brucei brucei | 6 μM (Meco-Navas et al. 2018) |
Salicylic hydroxamic acid | T. brucei brucei | 4 nM (Young et al. 2020) |
8-Hydroxyquinoline | P. falciparum | 11 μM (Roberts et al. 2004) |
8-Hydroxyquinoline | C. parvum | 0.7 μM (Roberts et al. 2004) |