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. 2025 Sep 12;16:1668173. doi: 10.3389/fimmu.2025.1668173

Table 2.

Outlines the mechanisms of action and effects of various compounds and pharmaceuticals on the AhR/IL-22 pathway.

Name Mechanism Result Reference
Chitooligosaccharides Restores the AHR-IL-22 pathway to normal, and promotes MUC2 expression Alleviates DSS-induced colitis in mice (94)
Akkermansia muciniphila Regulates Trp metabolism, activates AhR signaling and upregulates AhR target genes, such as IL-22 Reduces colon inflammation (91)
Atorvastatin Regulates intestinal flora imbalance, enhances microbial tryptophan metabolism, and increases AhR and IL-22 expression. Alleviates UC (88)
Dietary tryptophan supplementation Activates the AhR-mediated IL-22/Stat3 pathway Amelioration of DSS-induced colitis (86)
Fructo-oligosaccharides Regulates microbial tryptophan metabolism promotes the production of IAA and IPA, thereby triggering AhR/IL-22 axis activation Reduces symptoms of DSS-induced colitis (45)
Portulaca oleracea L-derived exosome-like nanoparticles Increasing the abundance of Lactobacillus reuteri and raising the levels of indole derivatives leads to the activation of AhR in conventional CD4+ T cells and increases IL-22 levels. Reduces UC in mice (87)
Lactiplantibacillus plantarum D266 Shaping the gut microbiota and Trp metabolism leads to activation of AhR and subsequent enhancement of IL-22 production Improvement of IBS symptoms (124)
Baicalein Upregulates CYP1A1 expression and promotes IL-22 production in ILC3 through activation of AhR Ameliorates symptoms and intestinal barrier function in UC mice (85)
Coptis chinensis polysaccharides
and Berberine
Boosts SCFA-producing bacteria, raising SCFA levels and activating the AhR/IL-22 pathway Improvement of symptoms in UC mice (89)
L-Fucose Stimulation of IL-22 secretion by CD4+ T cells in mouse splenocytes and ILC3 cells in LPMCs through activation of the nuclear AHR Improvement of symptoms in UC mice (48)
Fucoidan Decreases UC-induced AhR and IL-22 expression Treats with UC induced in rats (90)
6-formylindolo [3,2-b]carbazole AHR physiological activator, FICZ/AHR/CYP1A1 feedback regulation, stimulates IL-22 expression by a variety of different immune cells (including ILC3) Enhances the reinforcement of the intestinal epithelial barrier and aids in tissue repair, supporting intestinal balance. (62)
Lactobacillus rhamnosus GG Promotes ILC3 activation and IL-22 production through AhR interaction with ILC3s Prevention of virus enteric infections (13)
Hymenolepis nana antigens Enhances ISCs growth and development via the AhR/IL-22 pathway. Alleviating symptoms in UC mice (96)
Ganoderic acid A Regulation of intestinal flora and enhancement of AhR activity to promote IL-22 production Improvement of inflammatory bowel disease (115)
Infliximab Promotes IL-22+CD4+ T (Th22) cell differentiation in CD patients through AhR improves CD symptoms (113)
Dried ginger essential oil Regulation of intestinal microbiota and tryptophan metabolite IAA-AHR/IL-22/STAT3 signaling axis Alleviating 5-Fluorouracil-induced damage to the intestinal epithelial barrier in mice with mucositis (12)
Lactobacillus paracaseiL21 Activates the HIF1α/AhR pathway, increases IL-22 and mucins MUC2 to restore the goblet cell population Alleviates DSS-induced colitis (92)
Quercetin Increases IPA levels to activate the AhR/IL-22 pathway Reduces obesity and chronic intestinal inflammation (132)
Lactiplantibacillus plantarum producing high levels of indole-3-lactic acid Activates AHR signaling in the intestine by metabolizing tryptophan, activating downstream AHR signaling (such as CYP1A1, IL-22, and STAT3) to alleviate colitis Alleviates DSS-induced colitis in mouse models (93)