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. 2025 Oct 16;17(20):3337. doi: 10.3390/cancers17203337
ATAD2 ATPase family AAA domain-containing protein 2
BRD bromodomain
ANCCA AAA+ nuclear coregulator cancer-associated
CTA cancer-testis antigen
ES embryonic stem cells
Rb retinoblastoma
ERα estrogen receptor alpha
ATP adenosine Triphosphate
ADP adenosine diphosphate
DNA deoxyribonucleic acid
MD molecular dynamics
AIB1 amplified in breast cancer 1
RAC3 receptor-associated coactivator 3
TRAM1 translocation-associated membrane protein 1
E2 estradiol
ORF open reading frame
cAMP cyclic adenosine monophosphate
CBP CREB-binding protein
p300 EP300 or E1A binding protein p300
E2F early region 2 binding factor
c-Myc cellular myelocytomatosis
AKT protein kinase B
HIF1α hypoxia inducible factor 1 subunit alpha
GBM glioblastoma
MAPK mitogen-activated protein kinase
Asn asparagine
kDa kilodaltons
E2F1 early region 2 binding factor transcription factor 1
VCP valosin-containing protein
Hsp104 heat shock protein 104
NSF N-ethylmaleimide-sensitive factor
Arg arginine
Abo1 ATP-binding cassette subfamily F member 1
Pro proline
Val valine
MCM7 minichromosome maintenance complex 7
SRC-3 steroid receptor coactivator-3
RNA ribonucleic acid
CDK cyclin-dependent kinases
NCOA3 nuclear receptor coactivator
B-MYB B-Myeloid myeloblastosis
OS osteosarcoma
TNBC triple-negative breast cancer cells
Top2A DNA topoisomerase II alpha
DLGAP5 discs large-associated protein 5
Bub1 budding uninhibited by benzimidazole 1
MCM10 minichromosome maintenance protein 10
Kif kinesin family
NOL1 nucleolar protein 1
GPAT glycerol-3-phosphate acyltransferase
HSP60 heat shock protein 60
CAD carbamoyl-phosphate synthetase 2, aspartate transcarbamylase, and dihydroorotase
CDC25A cell division cycle 25A
AIM1 absent in melanoma 1
CCNE1 cyclin E1
ATR ataxia telangiectasia and Rad3-related protein
MLL1 mixed lineage leukemia protein-1
IRS-2 insulin receptor substrate 2
SNK serum-inducible protein kinase
AR androgen receptor
EZH2 enhancer of zeste homolog 2
PARP poly(ADP-ribose) polymerase
PC prostate cancer
HCC hepatocellular carcinoma
Bcl-2 B-cell leukemia/lymphoma 2 protein
MKK3/6 mitogen-activated protein kinase 3/6
PI3K phosphatidylinositol 3-kinases
mTOR mammalian target of rapamycin
pAKT phosphorylated protein kinase B
Miz1 c-Myc-interacting zinc finger protein-1
ESCC esophageal squamous cell carcinoma
SHH sonic hedgehog protein
SMO smoothened
GLUT1 glucose transporter type 1
HK2 hexokinase 2
GLI glioma-associated oncogene
EMT epithelial to mesenchymal transition
MMPs matrix metalloproteases
PTCH1 protein patched homolog 1
CRC colorectal cancer
OSCC oral squamous cell carcinoma
NF-κB nuclear factor kappa-light-chain-enhancer of activated B cells
NSD2 nuclear receptor binding SET domain protein 2
KAc acetyl-lysine
IC50 half-maximal inhibitory concentration
Ile isoleucine
BET bromodomain and extraterminal
RCSB research collaboratory for structural bioinformatics
PDB protein data bank
Kd equilibrium dissociation constant
TR-FRET time-resolved fluorescence resonance energy transfer
NEAT1_2 nuclear enriched abundant transcript 1, isoform 2
MM/GBSA molecular mechanics with generalized Born and surface area solvation
miRs microRNAs
UTR untranslated region
CENP centromeric protein
Tyr tyrosine
Phe phenylalanine
Glu glutamic acid
Asp aspartic acid
Ala alanine
Gly glycine
Br bromine
GC gastric cancer
TRIM25 tripartite motif-containing protein 25
miR-126-5p microRNA-126-5p
OC ovarian cancer
pChk phosphorylated checkpoint kinase
PTC papillary thyroid carcinoma
CD8Tex cluster of differentiation 8 T cell exhaustion
Trp tryptophan
Met methionine
SAR structure-activity relationship
HATs histone acetyltransferases
HDACs histone deacetylases
CRNDE colorectal neoplasia differentially expressed
PDAC pancreatic ductal adenocarcinoma