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. 2025 Apr 3;15(12):4601–4610. doi: 10.1007/s13346-025-01841-9

Table 2.

Pharmacokinetic parameters for cancellous bone 5 mm and 10 mm

Pharmacokinetic parameters 2 mL CarboCell 4 mL CarboCell Difference P-value
AUC0 − 24 h, min•µg/mL (95%CI)
Cancellous bone (5 mm) N = 8 202.7 (164.0; 641.3) N = 2 884.9 (407.7; 1362.2) 482.2 (-51.3; 1015.83) 0.071
Cancellous bone (10 mm) N = 8 475.0 (164.2; 785.7) N = 2 296.9 (-324.6; 918.5) -178.0 (-872.9; 516.9) 0.595
Cmax, µg/mL (95% CI)
Cancellous bone (5 mm) N = 8 0.7 (0.01; 1.4) N = 2 2.2 (0.8; 3.6) 1.5 (0.0001;3.0) 0.05
Cancellous bone (10 mm) N = 8 0.8 (0.2; 1.3) N = 2 0.3 (-0.8; 1.3) -0.5 (-1.7; 0.7) 0.384

Area under the curve from time 0 to 24 h (AUC0 − 24 h); Peak drug concentration (Cmax)

AUC0 − 24 h and Cmax are given as medians