| FGFR | Fibroblast growth factor receptor |
| FGF | Fibroblast Growth Factor |
| TKI | Tyrosine Kinase Inhibitor |
| SAR | Structure–Activity Relationship |
| IC50 | Half maximal inhibitory concentration |
| Kd | Dissociation constant |
| MD | Molecular Dynamics |
| ERK | Extracellular Signal-Regulated Kinase |
| MEK | Mitogen-Activated Protein Kinase Kinase |
| MAPK | Mitogen-Activated Protein Kinase |
| PI3K | Phosphoinositide 3-kinase |
| AKT | Protein Kinase B |
| TACC3 | Transforming Acidic Coiled-Coil containing protein 3 |
| TNBC | Triple-Negative Breast Cancer |
| NSCLC | Non-Small Cell Lung Cancer |
| HCT116 | Human colorectal carcinoma cell line |
| RT4 | Human bladder cancer cell line |
| SRB | Sulforhodamine B |
| ADME | Absorption, Distribution, Metabolism, and Excretion |
| CYP | Cytochrome P450 |
| hERG | Human Ether-à-go-go-Related Gene (potassium channel) |
| MS | Mass Spectrometry |
| HRMS | High-Performance Liquid Chromatography |
| UV | Ultraviolet |
| ESI | Electrospray Ionization |
| FAB | Fast Atom Bombardment |
| CLint | Intrinsic Clearance |
| SEM | Standard Error of the Mean |
| SD | Standard Deviation |
| EDC | 1-Ethyl-3-(3-dimethylaminopropyl)carbodiimmide |
| DMAP | 4-Dimethylaminopyridine |
| DIAD | Diisopropyl azodicarboxylate |
| DBU | 1,8-Diazabicyclo[5.4.0]undec-7-ene |
| PEt3 | Triethylphosphine |
| TBSCl | tert-Butyldimethylsilyl chloride |
| TBAF | Tetra-n-butylammonium fluoride |
| TBDPS | tert-Butyldiphenylsilyl |
| DPPA | Diphenylphosphoryl azide |
| TCDI | 1,1′-Thiocarbonyldiimidazole |
| DMSO | Dimethyl sulfoxide |
| ACN | Acetonitrile |
| EtOAc | Ethyl acetate |
| THF | Tetrahydrofuran |
| DMF | Dimethylformamide |
| MeOH | Methanol |