225Ac	Actinium-225
68Ga	Gallium-68
77Lu	Lutetium-177
LD	Linear dichroism
BSA	Bovine serum albumin
CH3CN	Acetonitrile
CPM	Counts per minute
Cu(OAc)2	Copper(II) acetate
CuCl2	Copper(II) chloride
DCM	Dichloromethane
DIPEA	N,N-diisopropylethylamine
DMSO	Dimethyl sulfoxide
DNA	Deoxyribonucleic acid
DSC	N,N′-Disuccinimidyl carbonate
EC50	Half-maximal effective concentration
EDC	1-(3-Dimethylaminopropyl)-3-ethylcarbodiimide hydrochloride
EMEM	Eagle’s minimum essential medium
ESI-Q-Tof	Electrospray ionization quadrupole time-of-flight
FBS	Fetal bovine serum
FDA	Food and Drug Administration
Fmoc	Fluorenylmethyloxycarbonyl
G4	G-quadruplex
HATU	O-(7-azabenzotriazol-1-yl)-N,N,N′,N′-tetramethyluronium hexafluorophosphate
HEK-293	Human embryonic kidney 293 cells
HEPES	4-(2-Hydroxyethyl)-1-piperazineethanesulfonic acid
HPLC	High-performance liquid chromatography
IC50	Half-maximal inhibitory concentration
iTLC	Instant thin-layer chromatography
ivDde	1-(4,4-Dimethyl-2,6-dioxocyclohexylidene)ethyl
LC/MS/MS	Liquid chromatography tandem mass spectrometry
LEEs	Low-energy electrons
LET	Linear energy transfer
LNCaP	Lymph Node Carcinoma of the Prostate
MBq	Megabecquerel
MBq/nmol	Megabecquerel per nanomole
mCRPC	Metastatic castration-resistant prostate cancer
MeOH	Methanol
NOTA	2,2′,2″-(1,4,7-triazacyclononane-1,4,7-triyl)triacetic acid
PBS	Phosphate-buffered saline
PCa	Prostate cancer
PEG	Polyethylene glycol
PET	Positron emission tomography
PSA	Prostate-specific antigen
PSMA	Prostate-specific membrane antigen
RLT	Radioligand therapy
RNA	Ribonucleic acid
ROS	Reactive oxygen species
RPMI-1640	Roswell Park Memorial Institute 1640 medium
Rt	Retention time
SD	standard deviation
SPPS	Solid-phase peptide synthesis
TACN	Triazacyclononane
TFA	Trifluoroacetic acid
TFE	Trifluoroethanol
TIPS	Triisopropylsilane
TP	Terpyridine–platinum