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. 2002 Apr;46(4):991–995. doi: 10.1128/AAC.46.4.991-995.2002

TABLE 5.

SI values of phosphonate nucleotides and alkoxyalkyl analogs in HFF cells

Compound VV
CV
EC50 (μM) CC50 (μM) SIa EC50 (μM) CC50 (μM) SIa
CDV 46.2 278 6 44.7 278 6.2
HDP-CDV 0.8 31 37 0.6 31 50
ODE-CDV 0.2 14.3 65 0.3 14.3 49
cCDV 50.6 >302 >6 48.3 >302 >6.2
HDP-cCDV 3.8 >100 >26 2.1 >100 >48
ODE-cCDV 1.1 47.8 43.4 0.5 47.8 88.5
a

SI = CC50/EC50; EC50s are from Table 2; CC50s are from Table 4.