Figure 3.
Clinical workflow for ferroptosis-targeted therapy in drug-resistant cancer: from initial diagnosis to treatment adjustment. Step 1 (Initial Tumor Diagnosis): Clarify cancer pathological classification and assess prior treatment history to determine drug-resistant status. Step 2 (Ferroptosis Sensitivity Biomarker Detection): Analyze three types of markers—molecular markers (ACSL4, GPX4, SLC7A11, TfR1), metabolic markers (PUFA-PL content, LIP levels), and immune markers (CD8+ T cell infiltration, PD-L1 expression)—using methods including pathological biopsy and imaging. Step 3 (Patient Stratification): Classify patients into the sensitive group (≥2 ferroptosis-sensitive markers + positive CD8+ T cell infiltration) or non-sensitive group (fewer than 2 sensitive markers or negative CD8+ T cell infiltration). Step 4 (Treatment Planning): Sensitive group receives ferroptosis inducers combined with immunotherapy (PD-1 inhibitors restore CD8+ T cell function, enhancing IFNγ-mediated ferroptosis); non-sensitive group undergoes preprocessing with epigenetic regulators (re-detect biomarkers post-preprocessing to switch to sensitive group if eligible). Step 5 (Delivery System & Safety Monitoring): Select nanocarriers for targeted drug delivery; monitor hematology (liver/kidney function), cardiotoxicity (myocardial enzymes), and iron overload (serum ferritin <1000 ng/mL). Step 6 (Efficacy Assessment & Adjustment): Continue the original plan if effective (CR/PR) and safe (recheck every 2 cycles); re-test biomarkers if ineffective (SD/PD); stop treatment and administer iron chelators for excessive toxicity (resume with 50% dose reduction after toxicity alleviation).
