| AMR | antimicrobial resistance |
| BBB | blood–brain barrier |
| CFU/mL | colony-forming units per milliliter |
| CNS | central nervous system |
| DMSO | Dimethyl sulfoxide |
| femA | factor essential for methicillin resistance A gene |
| femB | factor essential for methicillin resistance B gene |
| femX | factor essential for methicillin resistance X gene |
| Fu | Fraction unbound |
| LDH | lactate dehydrogenase |
| MDR-SA | multidrug-resistant S. aureus |
| MIC | minimum inhibitory concentration |
| NS | no significance |
| OD | optical density |
| PBP2a | Penicillin-Binding Protein 2a |
| PBS | phosphate-buffered saline |
| PG | peptidoglycan |
| CA | Calcein AM |
| PI | propidium iodide |
| SAR | structure–activity relationship |
| SEM | scanning electron microscopy |
| ±SEM | standard error of the mean |
| TSA | tryptone soy agar |
| WHO | World Health Organization |