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. 2026 Jan 29;65(3):465–477. doi: 10.1007/s40262-026-01618-4

Table 3.

Impact of dose on MTX pharmacokinetics and AKI

Variables MTX dose: ≤3.5 g/m2
N = 43
MTX dose: 8 g/m2
N = 37
P value
Age (years) 68.4 (59.2–76.6) 68.8 (61.4–73.7) 0.835
Sex (male) 33 (76) 21 (56) 0.0962
Protocol dose (g/m2) 2.6 (1.75–3.48) 6.0 (4.7–7.7) <0.0001
Total dose (g) 5.1 (3.4–6.9) 11.5 (9.1–13.75) <0.0001
Kidney parameters at baseline
 Serum creatinine (mg/dL) 0.90 (0.79–1.08) 0.89 (0.66–1.09) 0.365
 Cystatin C (mg/dL) 1.03 (0.86–1.17) 1.08 (0.90–1.23) 0.352
 Estimated kidney function (mL/min)
  CKD-EPI eGFRcreatinine 89.3 (71.4–96.3) 90.1 (68.2–102.8) 0.647
  CKD-EPI eGFRcystatin C 74.0 (60.7–89.7) 65.4 (56.0–85.1) 0.249
  CKD-EPI eGFRcreatinine-cystatin C 82.5 (69.3–96.5) 80.2 (63.8–95.4) 0.661
Albumin at baseline (mg/L) 3.9 (3.3–4.2) 3.8 (3.5–4.1) 0.850
Clearance of methotrexate (L/h) 11.9 (10.6–13.1) 11.4 (10.6–12.1) 0.307
Occurrence of any stage of AKI (N = 17) 13 (30)a 4 (11)a 0.054

aPercent of column total

AKI acute kidney injury, CKD-EPI Chronic Kidney Disease Epidemiology Collaboration, eGFR estimated glomerular filtration rate, MTX methotrexate