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. Author manuscript; available in PMC: 2026 Mar 11.
Published in final edited form as: J Clin Oncol. 2020 Aug 5;38(27):3217–3230. doi: 10.1200/JCO.20.01364

TABLE 2.

Study Outcomes: Efficacy of Larotrectinib in TRK Fusion-Positive Cancers in Adults and Children

Outcome Study Results Certainty of the Evidence (quality of evidence) Plain Text Summary
Overall response rate (primary outcome)a ORR: 75%a (95% CI, 61% to 85%; pre-established lower boundary of 30% ruled out); 13% complete response (95% CI, 6% to 25%); 62% partial response (95% CI, 49% to 75%); 13% stable disease (95% CI, 6% to 25%); 9% progressive disease (95% CI, 3% to 20%); 4% early withdrawal because of clinical deterioration (95% CI, 0.5% to 13.5%) Low (1, 2) Larotrectinib may improve overall response for patients with TRK fusion-positive tumors
Progression-free survival 55% progression-free at 1 year (95% CI, 42% to 67%) Low (1, 2) Larotrectinib may improve progression-free survival for patients with TRK fusion-positive tumors
Most common grade 3–4 adverse events 1,038 events occurred among 55 patients (93% grade 1 or 2; 7% grade 3 or 4): Very low (1) Larotrectinib may result in adverse events for patients with TRK fusion-positive tumors
Anemia (11%)
Increased level of ALT or AST (7%)
Weight increase (7%)
Decreased neutrophil count (7%)
Drug reductions or discontinuations 15% had dose reductions related to adverse events; no discontinuations as a result of drug-related adverse events were recorded Very low (1) Larotrectinib may result in dose reductions for patients with TRK fusion-positive tumors

NOTE. Results from Drilon et al.17 (1) Downgrade: commercially funded; indirectness: locally advanced included. (2) Upgrade: large magnitude of effect. Population: Fifty-five patients with TRK fusion-positive locally advanced or metastatic tumors, including 1 patient with pancreatic cancer. Intervention: Larotrectinib (20 patients treated in dose-escalation study and 35 treated at a therapeutic dose of 100 mg orally twice daily). Comparator: no comparator arm. ALT, alanine aminotransferase; AST, aspartate aminotransferase.

a

Independently assessed according to the RECIST version 1.1.19 Overall response rate: sum of complete and partial responses.19