2D	2-Dimensions
3D	3-Dimensions
ABC	ATP-Binding Domain
ADMET	Absorption, Distribution, Metabolism, Excretion, and Transport
ADP	Adenosine Diphosphate
ATCC	American Type Culture Collection
ATP	Adenosine Triphosphate
ATX	Chiral Aminated Thioxanthone
BINANA	BINding ANAlyzer
CAR	Constitutive androstane receptor
CNN	Convolutional neural network
CI	Confidence Interval
DBP	Drug-Binding Pocket
DBS	Drug-Binding Site
DMSO	Dimethyl sulfoxide
DNA	Deoxyribonucleic acid
EDTA	Ethylenediamine tetraacetic acid
FBS	Fetal Bovine Serum
FI	Fluorescence Intensity
FIIA	FI of RHO123 Inhibited Accumulation
FINA	FI of RHO123 Normal Accumulation
HBSS	Hank’s balanced salt solution
HK-2	Human Kidney 2
HPLC-DAD	High-Performance Liquid Chromatography—Diode Array Detection
IC50	Half-Maximal Inhibitory Concentration
ICH	Intracellular Coupling Helices
IUPAC	International Union of Pure and Applied Chemistry
MDR	Multidrug Resistance
MDR1	Multidrug Resistance 1
MFI	Mean Fluorescence Intensity
MOE	Molecular Operating Environment
MTT	3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyl tetrazolium bromide
NBD	Nucleotide Binding Domain
Nrf2	Nuclear factor erythroid 2-related factor 2
NR	Neutral Red
OX	Oxygenated Xanthone
PBS	Phosphate-Buffered Saline
P-gp	P-glycoprotein
PPAR	Peroxisome proliferator-activated receptor
PXR	Pregnane X receptor
RHO123	Rhodamine 123
RPMI	Roswell Park Memorial Institute
SMILES	Simplified Molecular Input Line Entry System
TMD	Transmembrane Domain
TMH	Transmembrane Helice
TX	Thioxanthone
X	Xanthone
ZOS	Zosuquidar