| AUC | Area under the curve |
| CL | Clearance |
| CYP | Cytochrome P450 |
| EHMT2 | Euchromatic histone-lysine N-methyltransferase 2 |
| GLP | G9a-like protein |
| H3K9me1/2 | Mono- and di-methylation of histone H3 Lys9 |
| HDMs | Histone demethylases |
| HMTs | Histone methyltransferases |
| i.p. | Intraperitoneal |
| IS | Internal standard |
| i.v. | Intravenous |
| LLOQ | Lower limit of quantification |
| MRT | Mean residence time |
| NK | Natural killer |
| PK | Pharmacokinetic |
| p.o. | Oral |
| TGI | Tumor growth inhibition |