| EA | Ethyl Acetate |
| TEA | Triethylamine |
| BBr3 | Boron Tribromide |
| LiHMDS | Lithium bis(trimethylsilyl)amide |
| DBU | 1,8-Diazabicyclo [5.4.0]undec-7-ene |
| p-TsOH | p-Toluenesulfonic Acid |
| TFA | Trifluoroacetic acid |
| PPA | Polyphosphoric Acid |
| MOM | methoxymethyl ether |
| DHP | 3,4-Dihydro-2H-pyran |
| PPTS | Pyridinium p-Toluenesulfonate |
| EDC | 1-(3-Dimethylaminopropyl)-3-ethylcarbodiimide (hydrochloride) |
| DMAP | 4-Dimethylaminopyridine |
| TBAB | Tetrabutylammonium bromide |
| DMF | N, N-Dimethylformamide |
| DEG | Diethylene glycol |
| LDA | Lithium diisopropylamide |
| TMSCl | Chlorotrimethylsilane |
| THF | Tetrahydrofuran |
| m-CPBA | meta-Chloroperoxybenzoic acid |
| BF3·OEt2 | Boron trifluoride etherate |
| PTT | phenyltrimethylammonium tribromide |
| Pd(PPh3)4 | Tetrakis(triphenylphosphine)palladium |
| i-PrOH | Isopropyl Alcohol |
| Py | pyridine |
| DEP | diethyl phosphite |
| DMS | dimethyl sulfate |
| Bi(OTf)3 | Bismuth(III) trifluoromethanesulfonate |
| NMP | N-Methyl-2-pyrrolidone |
| TsOMe | Methyl p-toluenesulfonate |
| TBHP | Tert-Butyl hydroperoxide |
| DMDO | Dimethyldioxirane |
| Oxone | potassium peroxymonosulfate |
| DFT | density functional theory |
| DMSO | Dimethyl Sulfoxide |
| MOMCl | Chloromethyl methyl ether |
| PhNEt2 | N, N-Diethylaniline |
| DIBAL-H | Diisobutylaluminium hydride |
| SAR | Structure–activity relationship |