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. 2026 Aug 28;18(9):1082. doi: 10.3390/pharmaceutics18091082
ALK anaplastic lymphoma kinase
ARA acid-reducing agent
AUC area under the concentration–time curve
BCL-2 B-cell lymphoma 2
BCRP breast cancer resistance protein (ABCG2)
BCS Biopharmaceutics Classification System
BID twice daily
BTK Bruton tyrosine kinase
CDK cyclin-dependent kinase
CLL chronic lymphocytic leukemia
Cmax maximum plasma concentration
CYP cytochrome P450
DDI drug–drug interaction
EGFR epidermal growth factor receptor
EMA European Medicines Agency
F oral bioavailability
FDA Food and Drug Administration
GI gastrointestinal
H2RA histamine H2-receptor antagonist
HER2 human epidermal growth factor receptor 2
HLA human leukocyte antigen
MATE multidrug and toxin extrusion
OATP organic anion transporting polypeptide
OCT organic cation transporter
PARP poly(ADP-ribose) polymerase
P-gp P-glycoprotein (ABCB1)
PK pharmacokinetics
PPI proton pump inhibitor
SmPC summary of product characteristics
TDM therapeutic drug monitoring
TKI tyrosine kinase inhibitor
TLS tumor lysis syndrome
UGT uridine diphosphate glucuronosyltransferase
VEGFR vascular endothelial growth factor receptor