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. 2026 Oct 6;16(46):60303–60321. doi: 10.1039/d6ra07915f

Table 4. Enzyme inhibitory effects of the E. elaterium extractsa.

Parts Solvents AChE (mg GALAE per g) BChE (mg GALAE per g) Tyrosinase (mg KAE per g) Amylase (mmol ACAE per g) Glucosidase (mmol ACAE per g)
Aerial parts EA 1.89 ± 0.19a 4.63 ± 0.07a 54.77 ± 3.75e 0.96 ± 0.02a na
Acetone na na 65.95 ± 2.50a 1.02 ± 0.07a na
Acetone/water 0.66 ± 0.01d 0.97 ± 0.07e 61.70 ± 0.29abc 0.29 ± 0.02e na
Water na 0.98 ± 0.07e 47.10 ± 0.33f 0.08 ± 0.01f na
Fruit peels EA 1.79 ± 0.15a 2.55 ± 0.42cd 59.54 ± 1.71cd 0.65 ± 0.03b 6.58 ± 0.09c
Acetone 1.86 ± 0.10a 3.37 ± 0.57bc 61.50 ± 0.81bc 0.60 ± 0.04bc na
Acetone/water 0.98 ± 0.04c 1.66 ± 0.15de 59.41 ± 0.14cd 0.30 ± 0.01e na
Water na 1.39 ± 0.13e 37.20 ± 0.61g 0.07 ± 0.01f na
Seeds EA 1.40 ± 0.05b 3.28 ± 0.58bc 55.56 ± 0.91de 0.66 ± 0.03b 5.66 ± 0.08d
Acetone 1.66 ± 0.05a 3.55 ± 0.56b 57.08 ± 0.74de 0.55 ± 0.03cd 6.98 ± 0.30b
Acetone/water 1.84 ± 0.11a 3.28 ± 0.34bc 64.82 ± 0.21ab 0.47 ± 0.01d 7.54 ± 0.23a
Water 1.76 ± 0.02a 2.82 ± 0.01bc 42.98 ± 0.03f 0.08 ± 0.01f na
a

The values are reported as mean ± SD of three parallel measurements. GALAE: galantamine equivalent; KAE: kojic acid equivalent; ACAE: acarbose equivalent; and na: not active. Different letters indicate significant differences between the tested extracts (p < 0.05).