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. 2005 Dec 28;6(13):246. doi: 10.1186/gb-2005-6-13-246

Table 3.

Proteins that physically interact with AP-2 transcription factors

Protein Description Domain of AP-2 proteins that interacts* Function of interaction Reference
APC Adenomatous polyposis coli tumor suppressor Basic region Inhibition of β-catenin/TCF/LEF-dependent transcription [16]
CITED2 Coactivator DD Transcriptional activation [69]
CITED4 Coactivator n.d. Transcriptional activation [70]
CDP CCAAT displacement protein DBD, DD Repression of the hamster histone H3.2 promoter [71]
DEK Oncoprotein, chromatin remodeling n.d. Transcriptional activation [72]
E1A Transforming protein of adenovirus DBD, DD Repression of AP-2 target genes [73]
c-Myc Oncoprotein Carboxyl terminus Impairment of Myc/Max DNA-binding and transactivation [14]
PARP PolyADP-ribose polymerase Carboxyl terminus Transcriptional activation [74]
PAX-6 Transcription factor n.d. Stimulation of gelatinase B activation [75]
PC4 Coactivator Transcriptional activation [24]
P300/CBP Coactivator Amino terminus Transcriptional activation [69]
p53 Tumor suppressor n.d. Augmentation of p53-dependent transcription [76]
RAP74 Subunit of transcription factor TFIIF Central region containing DBD Unknown [74]
Rb Retinoblastoma tumor suppressor Amino terminus Repression of the hamster histone H3.2 promoter; transcriptional activation of the E-cadherin gene [77,78]
SP1 Transcription factor Basic region Transcriptional activation of the ovine CYP11A1 gene [79]
SV40T Transforming protein of SV40 virus n.d. Blocks DNA binding of AP-2 protein [12]
UBC9 E2-conjugating enzyme DBD, DD Sumoylation [80]
WWOX Tumor suppressor Amino terminus PY motif Cytoplasmic localization PPPY motif [17]
YB-1 Transcription factor n.d. Stimulation of gelatinase A transcription [81]
YY1 Transcription factor DBD, DD Stimulation of the hamster histone H3.2 promoter [82]

*Abbreviations: DBD, DNA-binding domain; DD, dimerization domain; n.d., not determined. It is currently not entirely clear whether Rb binds AP-2 only via the amino terminus [78], or whether the DNA-binding domain is also necessary [77].