Table 2.
Activation | Desensitization | Deactivation | ||||
---|---|---|---|---|---|---|
τ (ms) | n | τ (ms) | n | τ (ms) | n | |
2-Me-5-HT | ||||||
WT | 259 ± 14 | 13 | 5653 ± 383 | 10 | 633 ± 38 | 14 |
D298A | 54 ± 6** | 11 | 3462 ± 223** | 14 | 101 ± 5** | 11 |
D298E | 298 ± 12* | 15 | 9730 ± 1352** | 8 | 879 ± 53** | 11 |
Dopamine | ||||||
WT | 543 ± 18 | 10 | 17967 ± 2575 | 9 | 184 ± 15 | 10 |
D298A | 48 ± 6** | 21 | 5685 ± 761** | 11 | 69 ± 4** | 7 |
D298E | 832 ± 70** | 14 | 23794 ± 2644 | 10 | 273 ± 17** | 9 |
All data are given as mean ±s.e.m.
P < 0.05
P < 0.01, compared to WT.