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. 2005;7(Suppl 5):S3–S12.

Table 3.

Comparison of Time to Achieve Castrate Levels for GnRH Agonists

GnRH Agonist % Castrate at Days 28–30
Leuprolide acetate for depot suspension
7.5 mg 94
22.5 mg 95
30 mg 94
Goserelin acetate implant
3.6 mg NR
10.8 mg NR
Triptorelin pamoate
3.75 mg 91.2
11.25 mg 97.7
Leuprolide acetate for injectable suspension
7.5 mg 94
22.5 mg 99
30 mg 96
Leuprolide acetate implant
65 mg 99
Histrelin acetate implant
50 mg 100

GnRH, gonadotropin-releasing hormone.