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. 2005 Jun 27;146(1):33–40. doi: 10.1038/sj.bjp.0706311

Table A1.

Receptors and ion channels with no binding affinity for W-212393 (IC50>1000 nM)

Adenosin A1 (human) Opioid κ (human)
Adrenergic α1, nonselective (human) Opioid δ (human)
Adrenergic α2, nonselective (human) Serotonin 5-HT1A (rat)
Adrenergic β1 (human) Serotonin 5-HT2 (human)
Adrenergic β2 (human) Serotonin 5-HT3 (human)
Adrenergic β3 (human) Serotonin 5-HT4 (guinea-pig)
Bradykinin B2 (human) Serotonin 5-HT5A (human)
Dopamine D1 (human) Serotonin 5-HT6 (human)
Dopamine D2 (human) Serotonin 5-HT7 (human)
Dopamine D3 (human) Sigma, nonselective (guinea-pig)
Dopamine D4.4 (human) Somatostatin sst1 (human)
Dopamine D5 (human) Dopamine transporter (human)
GABAA, agonist site (rat) Norepinephrine transporter (human)
GABAA, benzodiazepine, central (rat)  
GABAB, nonselective (rat) Calcium channel, L-type (rat)
Glucocorticoid (human) Calcium channel, N-type (rat)
Glutamate, nonselective (rat) Sodium channel, Site 1 (rat)
Histamine H1 (human) Potassium channel [KATP] (hamster)
Melatonin ML (MT), nonselective (chicken) Potassium channel [SKCa] (rat)
Muscarinic, nonselective, Central (rat)  
Neuropeptide Y1 (human)  
Nicotinic acetylcholine (human)