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. 2005 Jun 27;146(1):33–40. doi: 10.1038/sj.bjp.0706311

Table B1.

W-212393 had no effect on enzyme activity (IC50>10 μM)

ATPase, H+/K+ (rabbit)
Carbonic anhydrase (human)
Catechol-O-methyltransferase (COMT) (porcine)
Cyclooxygenase (COX-1) (human)
HMG-CoA reductase (rat)
Lipoxygenase (5-LO) (human)
Monoamine oxidase (MAO-A) (human)
Monoamine oxidase (MAO-B) (human)
Nitric oxide synthase, inducible (iNOS) (mouse)
Nitric oxide synthase, Neuronal (nNOS) (rat)
Phosphodiesterase (PDE1) (bovine)
Phosphodiesterase (PDE5) (human)
Phospholipase (PLA2-I) (porcine)
Phospholipase (PLC) (bacillus cereus)
Protein serine/threonine kinase (Ca2+/calmodulin-dependent II) (rat)
Protein serine/threonine phosphatase (calcineurin, PP2B) (human)
Protein serine/threonine kinase (p38α) (human)
Protein serine/threonine kinase (PKA), nonselective (bovine)
Protein serine/threonine kinase (PKC), nonselective (rat)
Protein tyrosine phosphatase (PTP1B) (human)
Tyrosine hydroxylase (rat)