Figure 13.
Alternative α-helical mimetics that antagonize Bcl-xL: (a) trispyridylamide 30 (Ki=2.3 μM) and (b) terephthalamide 31 (IC50=35.0 μM).
Alternative α-helical mimetics that antagonize Bcl-xL: (a) trispyridylamide 30 (Ki=2.3 μM) and (b) terephthalamide 31 (IC50=35.0 μM).