Table 1.

Percent inhibition of c-Src by linked binding elements at 1 μM

Entry	Compound mixture*	% inhibition of c-Src
1	[90, 273, n = 2–6]	89  ± 5
2	[73, 273, n = 2–6]	87  ± 6
3	[44, 273, n = 2–6]	83  ± 8
4	[39, 273, n = 2–6]	63  ± 11
5	[273, 273, n = 2–6]	43  ± 20
6	[90, 90, n = 2–6]	13  ± 7
7	[73, 73, n = 2–6]	7  ± 6
8	[44, 44, n = 2–6]	9  ± 4
9	[39, 39, n = 2–6]	7  ± 11

Percent inhibition of enzyme activity at an inhibitor concentration of 1 μM as determined by the percent phosphorylation of the tyrosine kinase peptide substrate (biotin-KVEKIGEGTYGVVYK), [ATP] = 125 μM. 

^*Compounds are denoted by listing the two linked binding elements followed by the linker length.