TABLE 5.
Relationship of MIC and in vivo efficacy in the mouse thigh model for NCE ABI-0043
| S. aureus strain | Mutation | MIC | Lowest ED (mg/kg)a | Lowest ED/MICa |
|---|---|---|---|---|
| 29213 | None | 0.002 | 0.06 | 30 |
| ABS-052 | A477→D | 0.5 | 10 | 20 |
| ABS-100 | H481→Y | 2 | >160 | >80 |
The lowest ED is the dose (mouse thigh) resulting in a 1-log difference in bacterial titer compared with placebo-treated animals.