Table 2.
Summary of agonist affinities of Y-family receptor subtypes. (NPY, neuropeptide Y; PP, pancreatic polypeptide; PYY, peptide YY (see also Berglund et al. 2003).)
receptor | high-affinity agonists | intermediate-affinity agonists | low-affinity agonists |
---|---|---|---|
Y1 | NPY, PYY, Leu31,Pro34NPY/PYY | NPY2-36, NPY3-36, NPY13-36 | PP |
Y2 (presynaptic) | NPY, PYY, PYY3-36 | Leu31,Pro34NPY/PYY | PP |
Y4 | PP, NPY, PYY, Leu31,Pro34NPY/PYY | NPY2-36 | NPY/PYY fragments PYY3-36 |
Y5 | NPY, PYY, NPY2-36, NPY3-36, PYY3-36, Leu31,Pro34NPY/PYY | PP, NPY13-36, PYY13-36 | NPY/PYY fragments |
y6 | non-functional in man |