Table 2.
Compound | DAT/NET ratio | DAT/SERT ratio | Selectivity |
---|---|---|---|
Cocaine | 0.0270 | 0.0856 | Nonselective |
RTI-126 | 0.0127 | 0.0261 | Nonselective |
RTI-112 | 0.0222 | 0.0762 | Nonselective |
RTI-150 | 0.0008 | 0.0018 | DAT selective |
RTI-336 | 0.0024 | 0.0007 | DAT selective |
RTI-171 | 0.0035 | 0.0002 | DAT selective |
RTI-177 | 0.0026 | 0.0005 | DAT selective |
Relative selectivity of binding to monoamine transporter ligands in rat tissue (Kuhar et al., 1999).