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. 2002 Aug;54(2):157–167. doi: 10.1046/j.1365-2125.2002.01614.x

Table 1.

Estimates of intrinsic clearance (µl min−1 pmol−1 CYP, r2) of tamoxifen to Z-4-OH-tam by supersomes expressing wild-type recombinant CYP450 isoform protein.

Expressed CYP450 isoform Intrinsic clearance (r2)
CYP2B6 2.91×10−2 (0.998)
CYP2C9 3.71×10−2 (0.992)
CYP2C19 3.93×10−2 (0.999)
CYP2D6 4.20×10−2 (0.991)