Table 3. Transactivation in TRAF-α and -β cells.
| Compound | TRAF-α EC50, nM | TRAF-β EC50, nM |
|---|---|---|
| T3 | 1.3 (100% agonism) | 3.5 (100% agonism) |
| KB-141 | 11.2 (101% agonism) | 3.4 (105% agonism) |
| Compound | TRAF-α EC50, nM | TRAF-β EC50, nM |
|---|---|---|
| T3 | 1.3 (100% agonism) | 3.5 (100% agonism) |
| KB-141 | 11.2 (101% agonism) | 3.4 (105% agonism) |