Table 2. Pharmacokinetic parameters for 13C-DHU in plasma.
Dose | Cmax (µg ml−1) | AUC12 h (µg h ml−1) | tmax (h) | λz (1 h−1) | t1/2 (h) |
---|---|---|---|---|---|
50 mg | 0.102 | 0.144 | 0.49 | 0.68 | 1.10 |
±0.050 | ±0.048 | ±0.15 | ±0.18 | ±0.34 | |
100 mg | 0.251 | 0.378 | 0.56 | 0.78 | 0.91 |
±0.094 | ±0.135 | ±0.18 | ±0.11 | ±0.14 | |
200 mg | 0.551 | 1.054 | 0.93 | 0.60 | 1.37 |
±0.255 | ±0.449 | ±0.50 | ±0.19 | ±0.74 |
Values: mean ± SD (n = 12).