Table 3. Pharmacokinetic parameters for 13C-DHU in plasma.
Dose | Cmax (µg ml−1) | AUC12 h (µg h ml−1) | tmax (h) | λz (1 h−1) | t1/2 (h) |
---|---|---|---|---|---|
50 mg | 0.023 | 0.006 | 0.46 | – | – |
±0.035 | ±0.014 | ±0.16 | – | – | |
100 mg | 0.076 | 0.034 | 0.50 | 1.17 | 0.87 |
±0.040 | ±0.042 | ±0.19 | ±0.88 | ±0.61 | |
200 mg | 0.149 | 0.126 | 0.82 | 1.12 | 1.05 |
±0.081 | ±0.105 | ±0.45 | ±0.67 | ±1.05 |
–, Not calculated. Values: mean ± SD (n = 12).