TABLE 2.
E2 target | Name or description | UniGene Hs cluster | Function | Repression (n-fold) |
---|---|---|---|---|
Mitosis | ||||
ANLN | Anillin | 62180 | Actin binding protein involved in cytokinesis | 0.22 |
BIRC5 | Survivin | 514527 | Inhibitor of apoptosis; senses kinetochore tension | 0.2 |
BUB1 | Homolog of mitotic checkpoint Saccharomyces erevisiae BUB1 | 469649 | Spindle assembly checkpoint; linked to genetic instability | 0.34 |
CCNB1 | Cyclin B1 | 23960 | Complexes with p34 cdc2 to form the mitosis promoting factor | 0.31 |
Cdc25C | Cell cycle division | 656 | M phase inducer phosphatase; activates cdc2 by dephosphorylation | 0.36 |
CDCA1 | Cell division cycle associated 1 | 234545 | Homolog of yeast Nuf2; component of the NDC80 kinetochore | 0.27 |
CDCA8 | Cell division cycle associated 8 | 524571 | Component of the chromosomal passenger complex | 0.34 |
CDKN2C | Cyclin-dependent kinase Inhibitor | 525324 | P18/INK4 inhibits cyclin/cyclin-dependent kinase complexes | 0.46 |
CENPA | Centromeric protein | 1594 | Component of modified nucleosome; interacts with Aurora A | 0.26 |
CENPF | Centromeric protein | 497741 | Kinetochore | 0.23 |
CHK1 | Checkpoint homolog | 24529 | Inhibits cdc25C; prevents activation of cyclinB/cdc2; DNA damage checkpoint | 0.44 |
CKS1 | Cdc28 protein kinase 1B | 374378 | Activates cdc20 transcription; substrate targeting subunit of the SCF ubiquitin ligase | 0.45 |
CKS2 | Cdc28 protein kinase | 83758 | Cdc2-associated protein (meiosis) | 0.41 |
DEPDC1B | DEP domain-containing protein 1B | 482233 | DEP-containing protein | 0.25 |
DIAPH3 | Diaphanous protein homolog 3 | 283127 | Binds to Rho and to profilin; involved in cytokinesis | 0.36 |
ECT-2 | Epithelial cell transforming 2 | 518299 | Oncogen; binds to Rhoa protein to activate mitosis (ortholog of Drosophila Pebble) | 0.33 |
FBXO Emi1 | F box only | 520506 | Interacts with cdc20 and inhibits the APC mitotic ubiquitin ligase | 0.37 |
HisH4F | Histone H4F | 247816 | Forms centromers with CENPA | 0.2 |
HURP (DLG7) | Hepatoma up-regulated | 77695 | Cell cycle regulator; up-regulated in G2/M | 0.22 |
KIF11 | Kinesin family member 11 | 8878 | Spindle assembly | 0.25 |
KIF22 | Kinesin member 22 | 119324 | Metaphase chromosome alignment | 0.42 |
KIF4A | Kinesin family member 4 | 279766 | Motor protein that translocates PRC1 | 0.33 |
LBR | Lamin B receptor | 435166 | Role in chromosome assembly | 0.39 |
MPHOSDH1 | M phase phosphoprotein | 240 | Kinesin-related protein; M-phase promoting factor | 0.25 |
NUP188 | Nucleoprotein | 308340 | 0.34 | |
NUP107 | Nucleoporin | 524574 | Nucleo-cytoplasmic trafficking; part of the nuclear pore and associated to the kinetochores | 0.44 |
NUSAP1 | Nucleolar and spindle associated protein 1 | 511093 | Involved in mitotic spindle organization | 0.29 |
PRC1 | Protein regulating cytokinesis | 567385 | Associated with mitotic spindles; associates with KIF4; organizes spindle midzone formation | 0.23 |
RACGAP1 | Rac GTPase activated protein | 505469 | Master regulator of initiation of cytokinesis | 0.32 |
SGOL1 | Shugoshin-like 1 | 105153 | Binds and stabilizes microtubules; localized to kinetochores | 0.35 |
SPBC25 | Kinetochore | 421956 | Component of the NDC80 kinetochore complex | 0.26 |
SPC24 | Spindle pole body 24 | 381225 | Component of the NDC80 kinetochore complex | 0.33 |
STK6 | Ser/Thr kinase 6 | 250822 | Aurora A is targeted to the spindle apparatus by TPX2 and regulates its activity | 0.34 |
STMN1 | Stathmin | 209983 | Sequesters tubulin in a ternary complex; role in depolymerization of mitotic microtubules | 0.28 |
TTK | TTK protein kinase | 169840 | MPS1L1, PYT, and ESK; required for normal centrosome duplication | 0.44 |
TMPO | Thymopoietin lamina-associated polypeptide | 11355 | Structural organization of the nucleus; postmitotic nuclear assembly | 0.35 |
TOPK | Mitotic protein kinase | 104741 | Mitotic Ser/Thr kinase related to mitogen-activated protein kinase kinase | 0.27 |
TPX2 | Targeting protein for Xklp2 | 244580 | Proliferating associated protein P100; associated with spindle pole and spindle | 0.30 |
Replication and DNA repair | ||||
BARD1 | BRCA1-associated ring domain 1 | 54089 | Implicated in BRCA1 tumor suppression and DNA repair | 0.36 |
CCNE2 | Cyclin E | 567387 | G1/S transition | 0.1 |
DCC1 | RFC alternative complex | 315167 | Primed loading of PCNA on gapped DNA; defective sister chromatin cohesion | 0.34 |
DTYMK | Thymidylate kinase | 471873 | DNA synthesis pathway catalyzes dMTP to dTDP | 0.45 |
HNRPA1 | Heterogenous nuclear ribonucleopreotein | 546261 | Interacts with Fen1 during Okazaki fragment maturation | 0.46 |
MCM4 | Minichromosome maintenance | 460184 | Replication licensing complex, loaded at the origins before initiation and essential for elongation | 0.47 |
MELK | Maternal embryonic leucine zipper kinase | 184339 | Implicated in stem cell renewal and cell cycle progression | 0.31 |
NBS1 | Nibrin | 492208 | Part of the DNA repair complex MRE11/RAD50 | 0.42 |
Pfs2 | GINS2 | 433180 | DNA replication complex GINS | 0.29 |
PRIM2A | Primase polypeptide A | 485640 | Polymerase that synthesizes small RNA primers (Okazaki) | 0.45 |
RFC3 | Replication factor C | 115474 | DNA clamp loading complex; necessary for elongation of primed DNA | 0.33 |
TREX2 | 3′ Repair exonuclease 2 | 170835 | DNA replication and DNA repair | 0.47 |
UNG | Uracyl-DNA glycosylase | 191334 | DNA replication and DNA repair | 0.3 |
USP1 | Ubiquitin specific protease | 35086 | Involved in DNA repair; Fanconi anemia pathway | 0.4 |
Cell proliferation | ||||
DHFR | Dihydrofolate reductase | 83765 | Required for synthesis of purines, thymidylic acid, and certain amino acids | 0.32 |
DEK | DEK oncogene | 110713 | Acute myeloma; oncogene | 0.46 |
DLEU2 | Deleted in lymphocytic leukemia | 508041 | Candidate tumor suppressor gene | 0.4 |
HMMR | Hyaluronan mediated motility receptor | 72550 | Involved in cell motility; may also be involved in cellular transformation and metastasis | 0.22 |
IGSF1 | Immunoglobin superfamily | 22111 | Role in cell adhesion | 0.4 |
ITGB3BP | Human beta 3 endonexin | 1741 | Coactivator of hormone receptors | 0.44 |
MLF1 | Myeloid leukemia factor 1 | 85195 | Oncoprotein; negative regulator of cell cycle | 0.47 |
NET1 | Neuroepithelila cell transforming gene | 25155 | Rho exchange factor | 0.44 |
RHOG | RAS homolog gene family G | 501728 | GTP-binding protein; activates RAC | 0.48 |
SHCBP1 | Shc SH2 domain protein | 123253 | Linking activated cell surface receptors to the Ras pathway | 0.32 |
SHMT1 | Serine hydroxy methyltransferase 1 | 513987 | Plays an essential role in nucleic acids biosynthesis | 0.24 |
SHMT2 | Serine hydroxy methyltransferase 2 | 75069 | Cytosolic; mitochondrial | 0.45 |
SRC | v-src sarcoma | 195659 | Protoncogene | 0.24 |
SYTL2 | Synaptotagmin-like protein | 369520 | Binds to Rab27; involved in vesicle trafficking | 0.42 |
THBS2 | Thrombospondin | 371147 | Inhibitor of tumor growth and angiogenesis | 0.32 |
Miscellaneous | ||||
ASF1B | Anti-silencing function | 26516 | Assembles nucleosome during nucleotide excision repair | 0.33 |
BCAT1 | Branched-chain amino transferase | 438993 | Direct target of c-Myc regulation | 0.42 |
CPSF1 | Cleavage polyadenylation specific factor | 493202 | Addition of poly(A) tail to mRNA | 0.43 |
DDX39 | DEAD box protein 39 | 311609 | ATP-dependent RNA helicase | 0.44 |
JUNB | JunB proto-oncogene | 25292 | Member of the AP1 transcription factor | 0.41 |
MNS1 | Meiosis-specific nuclear structural protein | 444483 | Meiosis | 0.42 |
NF-YB | Nuclear transcription factor Y | 84928 | Binding to the CCAAT motif | 0.41 |
RBL1 | Retinoblastoma-like; P107 | 207745 | Partner of E2F4/5 | 0.47 |
SMYD3 | Set and Mynd domain containing 3 | 567571 | Histone methyl transferase | 0.46 |
SNRPB | Splicing factor | 83753 | Knockout generates mitotic spindle defect; part of snRNP | 0.44 |
Known E2F target genes are in bold. Numbers given in the last column are levels of transcription in E2-expressing cells compared to GFP-expressing cells; underlining indicates that the gene is present more than once in the array.