Table 1.
Antibody | BoNT/A KD (M) | Domain specificity | In vitro neutralization (fold over control) |
---|---|---|---|
HuC25 | 4.5 × 10−11 | HC | 6.82* |
3D12 | 6.1 × 10−11 | HC | 3.02 |
S25 | 1.7 × 10−9 | HC | 1.85 |
9D8 | 1.2 × 10−9 | HN | ND |
ING2 | 9.6 × 10−12 | LC | ND |
ING1 | 3.1 × 10−10 | LC-HN | ND |
Solution KD of HuC25, 3D12, ING1, and ING2 were measured in a flow fluorimeter (KinExA) (ref. 22 and unpublished data). KD of S25 and 9D8 were measured using surface plasmon resonance (BIAcore) 25. In vitro neutralization was determined as time to 50% neuroparalysis in the mouse hemidiaphragm assay and is expressed as fold over control 17.
In vitro neutralization data for C25, murine precursor of humanized C25, HuC25.