Table 6.
Mean (% coefficient of variation) and median AUC(0,last) values for 3-OH-desloratadine by age group and dose
≥6 months−<1 year | ≥1 year−≤2 years | |||
---|---|---|---|---|
Parameter | 0.625 mg | 1.25 mg | 0.625 mg | 1.25 mg |
Mean AUC(0,last) (ng ml−1 h) | 9.29 (47) | 18.1 (71) | 6.30 (44) | 16.5 (65) |
Median AUC(0,last) (ng ml−1 h) | 7.30 | 16.4 | 5.85 | 15.6 |
Mean AUC(0,last) ratio (%) | 38.0 (55) | 51.8 (61) | 42.4 (58) | 64.1 (81) |
Median AUC(0,last) ratio (%) | 38.4 | 50.2 | 43.2 | 58.7 |
AUC(0,last) ratio = (AUC(3-OH-desloratadine) : AUC(desloratadine)) ×100.