Table 1.
Mean fu of indinavir (n = 2) and saquinavir (n = 2) in buffer solutions of HSA and/or AAG
fu | ||||
---|---|---|---|---|
Protein concentration (g l−1) in isotonic phosphate buffer | Indinavir1.00 mg l−1 | Indinavir8.00 mg l−1 | Saquinavir0.15 mg l−1 | Saquinavir1.50 mg l−1 |
HSA 20.0 | 0.73 | 0.62 | 0.035 | 0.020 |
HSA 30.0 | 0.64 | 0.60 | 0.026 | 0.019 |
HSA 40.0 | 0.66 | 0.59 | 0.011 | 0.014 |
AAG 0.20 | 0.81 | 0.82 | 0.070 | 0.14 |
AAG 0.60 | 0.74 | 0.68 | 0.016 | 0.017 |
AAG 2.00 | 0.34 | 0.26 | 0.0052 | 0.0073 |
HSA 30.0/AAG 0.20 | 0.68 | 0.58 | 0.0060 | 0.021 |
HSA 30.0/AAG 0.60 | 0.51 | 0.56 | 0.0065 | 0.015 |
HSA 30.0/AAG 2.00 | 0.29 | 0.31 | 0.0029 | 0.0038 |