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. 2006 Sep 19;63(3):315–321. doi: 10.1111/j.1365-2125.2006.02766.x

Table 1.

Mean fu of indinavir (n = 2) and saquinavir (n = 2) in buffer solutions of HSA and/or AAG

fu
Protein concentration (g l−1) in isotonic phosphate buffer Indinavir1.00 mg l−1 Indinavir8.00 mg l−1 Saquinavir0.15 mg l−1 Saquinavir1.50 mg l−1
HSA 20.0 0.73 0.62 0.035 0.020
HSA 30.0 0.64 0.60 0.026 0.019
HSA 40.0 0.66 0.59 0.011 0.014
AAG 0.20 0.81 0.82 0.070 0.14
AAG 0.60 0.74 0.68 0.016 0.017
AAG 2.00 0.34 0.26 0.0052 0.0073
HSA 30.0/AAG 0.20 0.68 0.58 0.0060 0.021
HSA 30.0/AAG 0.60 0.51 0.56 0.0065 0.015
HSA 30.0/AAG 2.00 0.29 0.31 0.0029 0.0038