Table 2.
Some compounds that modulate ABCG2 activitya
| Endogenous modulators | Dietary modulators | Exogenous modulators |
|---|---|---|
| Oestrone | Apigenin | FTC |
| 17 β-Oestradiol | Biochanin A | Ko143, Ko132 and Ko134 |
| Chrysin | GF120918 | |
| Genistein | Novobiocin | |
| Hesperetin | Tamoxifen | |
| Kaempferol | Toremifene | |
| Naringenin | TAG 139, TAG 11 | |
| Silymarin | Gefitinib | |
| Folate | Imatinib mesylate | |
| Flavopiridol |
Abbreviation: FTC, fumitremorgin C.
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