Table 9.
AMAI Treatment
Treatment | Results | Effects |
Maximum agonism of mAR | ↑apoptotic proteins ↓bcl-2 (BC only) ↑bcl-2 (PC only) ↓AS3 ↑Ca++ influx |
↑ RD ↑ RD ↓ RD ↑ RG ↑ RD |
Maximum agonism of iAR | ↓apoptotic proteins ↓bcl-2 ↑AS3 ↓Ca++ influx ↑calreticulin |
↓ RD ↑ RD ↓ RG ↓ RD ↓ RD |
Maximum antagonism of ER-α | ↓bcl-2 | ↑ RD |
Maximum agonism of ER-β | ↓bcl-2 | ↑ RD |
Maximum antagonism of mER | ↓bcl-2 | ↑ RD |
Maximum antagonism of PRA | ↓bcl-2 | ↑ RD |
Maximum agonism of PRB | ↓bcl-2 | ↑ RD |
Maximum agonism of mPR | ↓bcl-2 | ↑ RD |
Maximum calcitriol | ↑AS3 ↑kill mitochondria |
↓ RG ↑ RD |