Table A2.
Partition coefficients for R- and S-ket and R- and S-nor
Parameter name | Value | Partition coefficient (unitless) |
---|---|---|
ppF | 332 | For ketamine (R or S) between blood and fat |
ppS | 4.83 | For ketamine (R or S) between blood and slowly perfused tissue |
ppR | 35.3 | For ketamine (R or S) between blood and rapidly perfused tissue |
ppK | 31.4 | For ketamine (R or S) between blood and kidney |
ppL | 16.7 | For ketamine (R or S) between blood and liver |
ppX | 10 | For ketamine (R or S) between blood and lung |
pmF | 1 | For norketamine (R or S) between blood and fat |
pmS | 1 | For norketamine (R or S) between blood and slowly perfused tissue |
pmR | 1 | For norketamine (R or S) between blood and rapidly perfused tissue |
pmK | 1 | For norketamine (R or S) between blood and kidney |
pmL | 1 | For norketamine (R or S) between blood and liver |
pmX | 1 | For norketamine (R or S) between blood and lung |