Table A2.
Partition coefficients for R- and S-ket and R- and S-nor
| Parameter name | Value | Partition coefficient (unitless) |
|---|---|---|
| ppF | 332 | For ketamine (R or S) between blood and fat |
| ppS | 4.83 | For ketamine (R or S) between blood and slowly perfused tissue |
| ppR | 35.3 | For ketamine (R or S) between blood and rapidly perfused tissue |
| ppK | 31.4 | For ketamine (R or S) between blood and kidney |
| ppL | 16.7 | For ketamine (R or S) between blood and liver |
| ppX | 10 | For ketamine (R or S) between blood and lung |
| pmF | 1 | For norketamine (R or S) between blood and fat |
| pmS | 1 | For norketamine (R or S) between blood and slowly perfused tissue |
| pmR | 1 | For norketamine (R or S) between blood and rapidly perfused tissue |
| pmK | 1 | For norketamine (R or S) between blood and kidney |
| pmL | 1 | For norketamine (R or S) between blood and liver |
| pmX | 1 | For norketamine (R or S) between blood and lung |