Table 1.
0.5 mg kg−1 | 1 mg kg−1 | 10 mg kg−1 | 30 mg kg−1 | |
---|---|---|---|---|
CL (ml min−1 kg−1) | 1.92 ± 0.20 | 2.12 ± 0.07 | 1.52 ± 0.12 | 1.00 ± 0.08 |
Vss (1 kg−1) | 0.42 ± 0.06 | 0.48 ± 0.08 | 0.44 ± 0.04 | 0.42 ± 0.14 |
λz (min−1) | 0.0045 ± 0.00046 | 0.0038 ± 0.00077 | 0.0031 ± 0.00044 | 0.0022 ± 0.0008 |
MRT (min) | 222 ± 43 | 240 ± 45 | 305 ± 32 | 423 ± 158 |
AUC (mg min ml−1) | 0.24 ± 0.03 | 0.46 ± 0.16 | 6.0 ± 0.5 | 28 ± 3 |
Data are mean ± SEM, with five animals per dose group.