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. Author manuscript; available in PMC: 2008 Dec 1.
Published in final edited form as: Bioorg Med Chem Lett. 2007 Sep 15;17(23):6638–6642. doi: 10.1016/j.bmcl.2007.09.048
Route t1/2 (hr) AUC∞ (μg hr/L) Volume of distribution (L/kg) Clearance (L/hr/kg) Bio-availability

IV (10mg/kg) 2.6 19091 2.0 0.53 N/A
Oral (100 mg/kg) 4.2 65931 9.3 1.58 34.5%