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. Author manuscript; available in PMC: 2008 Dec 24.
Published in final edited form as: Tetrahedron Lett. 2007 Dec 24;48(52):9140–9143. doi: 10.1016/j.tetlet.2007.10.119

Table 1.

Inline graphic
Reactant Product R Yield (%)*
4a 3a m-CF3 62%
4b 3b H 66%
4c 3c o-OCH3 69%
4d 3d p-OCH3 67%
4e 3e p-CH3 61%
4f 3f p-tbutyl 64%
4g 3g o-F 60%
4h 3h p-F 66%
4i 3i 3,5-CF3 42%
4j 3j o-OCH3, 5-F 66%
4k 3k 3,5-F 51%
4l 3l m-NO2 58%
4m 3m m-NO2, p-CH3 59%
4n 3n o-Cl 59%
*

Yields calculated from intermediate 2 following the one-pot Suzuki coupling and Boc deprotection