Official websites use .gov
A
.gov website belongs to an official
government organization in the United States.
Secure .gov websites use HTTPS
A lock (
) or https:// means you've safely
connected to the .gov website. Share sensitive
information only on official, secure websites.
Inhibition of 20S proteasome by intra-ring bivalent inhibitors, IC50, μM
| Inhibitor | PGPH | Trypsin-like | Chymotrypsinlike |
|---|---|---|---|
| Ac-LLnL-H (1) | >100 | >100 | 2.1 |
| OHC-CO-LGPGGLLnL-H (3) | >100 | >100 | 0.08 |
| Lev-KKGEVSLE-H (4) | 102 | >100 | >100 |
| Saa-KKGEVSLE-H (5) | 82 | >100 | >100 |
| Saa-AAEVSLE-H (6) | 146 | >100 | >100 |
Lev, levulinic acid; Saa, 4-oxobutyric acid.
